Basic Information
ID: ALA3795791
Type: Binding
Description: Inhibition of KDM5A (unknown origin) using substrate peptide/ascorbate/2-OG/ Fe(2) as substrate at 10 uM preincubated for 15 mins followed by addition of substrate peptide/ ascorbate/2-OG/ Fe(2) measured after 1 hr by AlphaLISA method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3795791
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 317.32 | 1.60 | 1.60 |
| 299.33 | 1.46 | 1.46 |
| 232.22 | 1.77 | 1.77 |
| 248.67 | 2.28 | 2.28 |
| 214.23 | 1.63 | 1.63 |
| 228.25 | 1.94 | 1.94 |
| 258.24 | 1.33 | 1.33 |
| 154.13 | -0.54 | -0.54 |
| 242.24 | 1.62 | 1.62 |
| 232.20 | 1.21 | 1.21 |
| 195.23 | -0.40 | -0.40 |
| 128.11 | -0.10 | -0.10 |
| 144.56 | 0.42 | 0.42 |
| 110.12 | -0.24 | -0.24 |
| 124.15 | 0.07 | 0.07 |
| 178.12 | 0.78 | 0.78 |
| 213.22 | -0.26 | -0.26 |
| 202.22 | 1.55 | 1.55 |
| 220.21 | 1.69 | 1.69 |
| 232.24 | 1.56 | 1.56 |
| 230.23 | 1.13 | 1.13 |
| 271.24 | 1.29 | 1.29 |
| 160.18 | 0.92 | 0.92 |