Assay Report Card

Basic Information

ID: ALA3796231

Type: Binding

Description: Inhibition of chymotrypsin like activity of human 20S proteasome using Suc-Leu-Leu-Val-Tyr-AMC as substrate preincubated for 10 mins followed by substrate addition measured after 1 hr by spectrofluorimetric analysis

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
384.25
436.25
436.36
436.36
518.47
620.64
620.64
566.51
570.47
570.58
570.58
570.58
570.58
604.60
618.63
622.59
522.54
536.57
536.57
620.64
609.62
570.58
604.60
618.63
536.57
522.54
570.58
620.64
616.61
620.64
454.42
454.42
502.46
528.50
562.52
478.48
512.50
526.53
585.55
633.60
398.27
452.24
519.16
587.15
511.21