Assay Report Card

Basic Information

ID: ALA3801641

Type: Binding

Description: Inhibition of human poly His-tagged WDR5 (1 to 334 residues) interaction with MLL1 assessed as displacement of fluorescein isothiocyanate labelled 9-Ala-FAM peptide substrate from WDR5 expressed in Escherichia coli BL21(DE3)-V2R-pRARE2 cells by fluorescence polarization assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
425.372.312.31
498.514.004.00
507.524.614.61
495.514.554.55
555.603.903.90
514.513.423.42
472.473.043.04
471.483.653.65
559.592.592.59