Basic Information
ID: ALA3803119
Type: Binding
Description: Inhibition of full length N-terminal His-tagged SMYD3 (1 to 428 residues) (unknown origin) expressed in Escherichia coli using N-terminal GST-tagged MEKK2 as substrate preincubated for 30 mins followed by substrate addition by scintillation proximity assay in presence of [3H]SAM
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3803119
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 259.31 | 0.66 | 0.66 |
| 380.47 | 0.05 | 0.05 |
| 414.92 | 0.71 | 0.71 |
| 420.54 | 0.70 | 0.70 |
| 446.57 | 1.24 | 1.24 |
| 481.02 | 1.89 | 1.89 |
| 460.60 | 1.58 | 1.58 |
| 460.60 | 1.26 | 1.26 |
| 591.10 | 3.94 | 3.94 |
| 539.10 | 1.98 | 1.98 |
| 481.02 | 1.89 | 1.89 |
| 481.02 | 1.89 | 1.89 |
| 446.57 | 1.51 | 1.51 |
| 482.01 | 1.23 | 1.23 |
| 496.03 | 1.49 | 1.49 |
| 510.06 | 1.83 | 1.83 |
| 572.13 | 3.06 | 3.06 |
| 465.55 | 0.71 | 0.71 |
| 461.59 | 0.88 | 0.88 |
| 447.56 | 0.57 | 0.57 |