Basic Information
ID: ALA3803248
Type: Binding
Description: Inhibition of recombinant rat N-terminal GST-tagged DYRK1A (1 to 499 residues) expressed in Escherichia coli using KKISGRLSPIMTEQ-NH2 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control
Format: BAO_0000019
Organism: Rattus norvegicus
Target: Dual specificity tyrosine-phosphorylation-regulated kinase 1A(ALA5508)
Document: ALA3797082
Inhibition of recombinant rat N-terminal GST-tagged DYRK1A (1 to 499 residues) expressed in Escherichia coli using KKISGRLSPIMTEQ-NH2 as substrate at 100 uM incubated for 10 mins by scintillation counting method relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3803248
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 277.33 | 3.78 | 3.78 |
| 291.35 | 4.00 | 4.00 |
| 277.33 | 3.69 | 3.69 |
| 383.45 | 2.16 | 2.16 |