Assay Report Card

Basic Information

ID: ALA3803506

Type: Binding

Description: Inhibition of human Nav1.7 expressed in HEK293 cells assessed as inward peak current by ion-works quattro patch clamp electrophysiology method

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
4029.89
4087.93
3997.80
4013.78
3988.79
4016.80
4031.82
4047.86
4029.89
4030.87
4016.80
3988.79
4047.86
4030.87
4031.82
4045.84
4057.90
3988.79
3958.76
3981.80
4045.84
3997.80
4144.98
4139.94
4128.98
4101.91
4101.91
4074.84
4172.00
4123.96
4107.96
4084.92
4133.99
4157.98
4157.03
4157.03
4156.05
4157.98
4123.96
4214.08
4156.05
4112.94
4160.98
4096.94
4131.94
4122.97
4159.01
4160.98
4146.95
4146.01
4103.92
4146.01
4145.02
4163.00
4146.95
4128.91
4112.94
4203.06
4145.02
4260.11
4202.07
4054.90
4102.94
4038.90
4015.86
4064.93
4100.97
4045.88
4102.94
4087.97
4104.96
4045.88
4087.97
4086.99
4088.91
4045.88
4070.87
4145.02
4088.91
4086.99
4202.07
4230.09
4082.91
4130.95
4066.91
4101.91
4043.87
4130.95
4115.98
4132.97
4101.91
4115.98
4115.00
4116.93
4101.91
4098.89
4082.91
4173.04
4116.93
4115.00
4230.09
4203.01
4055.84
4103.88
4039.84
4074.84
4016.80
4065.87
4046.82
4115.94
4103.88
4088.91
4046.82
4074.84
4088.91
4087.93
4105.90
4089.85
4074.84
4046.82
4071.81
4055.84
4145.96
4087.93
4203.01
4016.80
4016.80
4007.84
4043.87
4074.84
4075.83
4107.92
4097.88
4073.90
4091.94
4047.82
4061.84
4059.87
4123.91
4151.92
4108.90
4074.88
4065.87
4101.95
4073.94
4060.81
4073.85
4129.97
4101.95
4115.94
3958.81
4074.88
3926.72
3827.59
3664.41
4144.98
4031.82
4092.95
4260.11
4089.85