Basic Information
ID: ALA3806630
Type: Binding
Description: Inhibition human full length PI3Kdelta catalytic subunit/p85alpha assessed as formation of PIP3 after 30 mins by europium labeled GRP-based TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3806630
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 417.86 | 3.88 | 3.88 |
| 392.85 | 3.58 | 3.58 |
| 377.83 | 4.00 | 4.00 |
| 402.85 | 3.87 | 3.87 |
| 417.86 | 3.46 | 3.46 |
| 416.87 | 4.06 | 4.06 |
| 417.86 | 3.46 | 3.46 |
| 435.88 | 2.68 | 2.68 |
| 460.85 | 4.60 | 4.60 |
| 452.40 | 2.80 | 2.80 |
| 459.42 | 2.53 | 2.53 |
| 406.88 | 3.89 | 3.89 |
| 422.88 | 3.59 | 3.59 |
| 416.87 | 3.57 | 3.57 |
| 492.97 | 4.98 | 4.98 |
| 493.96 | 4.38 | 4.38 |
| 494.95 | 3.77 | 3.77 |
| 494.95 | 3.77 | 3.77 |
| 511.95 | 4.52 | 4.52 |
| 482.94 | 3.71 | 3.71 |
| 418.87 | 3.46 | 3.46 |
| 432.88 | 3.04 | 3.04 |
| 452.31 | 4.11 | 4.11 |
| 442.31 | 3.82 | 3.82 |
| 452.31 | 4.11 | 4.11 |
| 431.89 | 3.76 | 3.76 |
| 450.87 | 3.18 | 3.18 |
| 450.87 | 3.18 | 3.18 |
| 467.32 | 3.69 | 3.69 |
| 457.89 | 2.91 | 2.91 |
| 462.90 | 3.05 | 3.05 |
| 500.87 | 4.06 | 4.06 |
| 496.91 | 3.85 | 3.85 |
| 482.88 | 3.98 | 3.98 |
| 482.90 | 2.78 | 2.78 |
| 517.33 | 4.63 | 4.63 |
| 468.86 | 3.32 | 3.32 |
| 486.85 | 3.46 | 3.46 |
| 434.41 | 2.66 | 2.66 |
| 452.40 | 2.80 | 2.80 |
| 452.40 | 2.80 | 2.80 |