Assay Report Card

Basic Information

ID: ALA3811916

Type: Binding

Description: Substrate activity at human LAT1 expressed in HEK cells assessed as efflux rate of [3H]-gabapentin at 200 uM after 5 to 180 secs by scintillation counting based trans-stimulation assay

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
183.180.780.78
181.190.350.35
165.190.640.64
131.170.440.44
241.292.312.31
174.20-1.34-1.34
307.090.950.95
179.220.950.95
179.220.950.95
199.641.291.29
199.180.490.49
244.091.401.40
291.091.251.25
193.251.201.20
207.271.761.76
221.301.941.94
255.322.232.23
215.641.001.00
260.091.111.11
195.220.660.66
209.250.910.91
223.271.471.47
237.301.641.64
271.321.941.94
257.292.012.01
209.250.960.96
179.220.950.95