Basic Information
ID: ALA3821343
Type: Binding
Description: Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane assessed as radioligand binding at 10 uM by microbeta scintillation counting method relative to control
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA3821343
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 229.63 | -1.08 | -1.08 |
| 311.78 | 0.72 | 0.72 |
| 333.78 | 0.99 | 0.99 |
| 282.70 | -0.34 | -0.34 |
| 328.81 | 0.09 | 0.09 |
| 319.76 | 0.95 | 0.95 |
| 320.74 | 0.34 | 0.34 |
| 362.83 | 0.54 | 0.54 |
| 301.69 | -0.78 | -0.78 |
| 426.89 | 0.03 | 0.03 |
| 287.67 | -1.17 | -1.17 |
| 337.75 | 1.09 | 1.09 |
| 379.88 | 1.68 | 1.68 |
| 411.88 | 0.36 | 0.36 |
| 329.75 | -0.30 | -0.30 |
| 325.72 | -1.50 | -1.50 |
| 320.74 | 0.34 | 0.34 |
| 382.26 | 0.71 | 0.71 |
| 384.27 | 1.09 | 1.09 |
| 404.69 | 1.43 | 1.43 |
| 439.13 | 2.09 | 2.09 |
| 449.14 | 1.54 | 1.54 |
| 415.24 | 0.69 | 0.69 |
| 463.80 | 0.49 | 0.49 |
| 400.27 | 0.79 | 0.79 |
| 400.27 | 0.79 | 0.79 |
| 430.30 | 0.80 | 0.80 |
| 414.25 | 0.51 | 0.51 |
| 491.86 | 1.18 | 1.18 |
| 503.87 | 1.35 | 1.35 |
| 442.35 | 1.96 | 1.96 |
| 553.93 | 2.36 | 2.36 |
| 454.24 | 1.68 | 1.68 |
| 347.81 | 1.17 | 1.17 |