Assay Report Card

Basic Information

ID: ALA3821346

Type: Binding

Description: Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane assessed as radioligand residence time at 10 uM by microbeta scintillation counting method (Rvb = 2.8 +/- 0.4 mins)

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
311.780.720.72
400.270.790.79
400.270.790.79
414.250.510.51
491.861.181.18