Assay Report Card

Basic Information

ID: ALA3821475

Type: Binding

Description: Displacement of [3H]ZM-241,385 from human N-terminal FLAG-tagged adenosine A2A receptor W246A 6.48 mutant expressed in HEK293 cell membrane assessed as decrease in radioligand residence time at 10 uM by microbeta scintillation counting method relative to control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
311.780.720.72
400.270.790.79
400.270.790.79
414.250.510.51
491.861.181.18