Basic Information
ID: ALA3829452
Type: Binding
Description: Inhibition of human ERAP1 preincubated for 30 to 60 mins followed by addition of Leu-AMC as substrate measured for 15 mins by spectrofluorimetric method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3829452
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 167.15 | 0.49 | 0.49 |
| 167.15 | 0.49 | 0.49 |
| 361.38 | 3.12 | 3.12 |
| 377.38 | 2.82 | 2.82 |
| 361.38 | 3.12 | 3.12 |
| 215.19 | 1.08 | 1.08 |
| 215.19 | 1.08 | 1.08 |
| 389.43 | 3.73 | 3.73 |
| 406.38 | 3.03 | 3.03 |
| 377.38 | 2.82 | 2.82 |
| 377.38 | 2.82 | 2.82 |
| 391.40 | 2.61 | 2.61 |
| 362.37 | 2.51 | 2.51 |
| 362.37 | 2.51 | 2.51 |
| 389.43 | 3.73 | 3.73 |
| 390.42 | 2.58 | 2.58 |
| 390.42 | 2.58 | 2.58 |
| 208.20 | -0.07 | -0.07 |
| 210.17 | -1.22 | -1.22 |
| 286.27 | 0.44 | 0.44 |
| 328.35 | 1.48 | 1.48 |
| 342.38 | 1.73 | 1.73 |
| 368.41 | 2.41 | 2.41 |
| 382.44 | 2.80 | 2.80 |
| 420.45 | 2.33 | 2.33 |
| 140.08 | -1.59 | -1.59 |
| 154.11 | -1.33 | -1.33 |
| 182.16 | -0.55 | -0.55 |
| 224.24 | 0.62 | 0.62 |
| 183.15 | -2.00 | -2.00 |
| 211.20 | -1.40 | -1.40 |
| 222.22 | 0.37 | 0.37 |
| 236.25 | 0.76 | 0.76 |
| 237.24 | -0.69 | -0.69 |
| 224.20 | -0.78 | -0.78 |
| 237.24 | -0.96 | -0.96 |
| 252.25 | -2.06 | -2.06 |
| 230.20 | 0.24 | 0.24 |
| 244.23 | 0.80 | 0.80 |
| 286.31 | 1.54 | 1.54 |
| 244.23 | 0.28 | 0.28 |
| 245.22 | -0.18 | -0.18 |
| 260.23 | 0.25 | 0.25 |
| 259.25 | -0.30 | -0.30 |
| 274.26 | 0.29 | 0.29 |
| 391.41 | 1.97 | 1.97 |
| 391.41 | 1.97 | 1.97 |