ID: ALA3830584
Type: Binding
Description: Inhibition of synthetic fluorescent ligand binding to recombinant truncated 6H-Flag-TEV-BRPF1 (622 to 738 residues) (unknown origin) expressed in Escherichia coli BL21 (DE3) cells after 30 mins by TR-FRET assay
Organism: Homo sapiens
Cell type: BL21-DE3
Bioactivity
Activity Types for Assay ALA3830584
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
380.45 | 2.74 | 2.74 |
341.37 | 2.15 | 2.15 |
325.37 | 2.45 | 2.45 |
354.41 | 2.20 | 2.20 |
369.42 | 2.93 | 2.93 |
399.45 | 2.29 | 2.29 |
412.45 | 1.78 | 1.78 |
426.52 | 2.86 | 2.86 |
394.43 | 2.82 | 2.82 |
413.47 | 2.94 | 2.94 |
440.50 | 2.38 | 2.38 |
438.53 | 3.00 | 3.00 |
220.27 | 1.66 | 1.66 |
277.32 | 1.62 | 1.62 |
305.38 | 2.40 | 2.40 |
332.40 | 1.21 | 1.21 |
347.42 | 2.03 | 2.03 |
339.40 | 2.92 | 2.92 |
340.38 | 2.31 | 2.31 |
340.38 | 2.31 | 2.31 |
340.38 | 2.31 | 2.31 |
341.37 | 1.71 | 1.71 |
370.41 | 2.32 | 2.32 |
370.41 | 2.32 | 2.32 |
399.45 | 2.93 | 2.93 |
399.45 | 2.38 | 2.38 |
395.46 | 1.55 | 1.55 |
409.49 | 1.89 | 1.89 |
394.48 | 2.60 | 2.60 |
392.46 | 2.51 | 2.51 |
394.48 | 3.13 | 3.13 |
394.48 | 3.13 | 3.13 |
409.49 | 1.94 | 1.94 |
409.49 | 1.94 | 1.94 |
409.49 | 1.94 | 1.94 |
409.49 | 1.94 | 1.94 |
437.54 | 2.35 | 2.35 |