Assay Report Card

Basic Information

ID: ALA3854797

Type: Binding

Description: Activation of recombinant human AMPK alpha1/beta2/gamma1 assessed as protection from Thr172 residue dephosphorylation up to 40 uM preincubated for 15 mins followed by incubation with PP2a for 60 mins measured 60 mins post okadaic acid/Cy5-labelled SAMS and ATP addition by TR-FRET assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
387.443.703.70