Basic Information
ID: ALA3858378
Type: Binding
Description: Displacement of [3H]-(S)-7-(2-chloro-3-(trifluoromethyl)benzyl)-6-methyl-3-(pyrazin-2-yl)-6,7-dihydro-[1,2,4]triazolo[4,3-a]pyrazin-8(5H)-one from recombinant human P2X7 receptor expressed in human 1321N1 cell membranes after 1 hr
Organism: Homo sapiens
Cell type: 1321-N1
Activity Charts
Bioactivity
Activity Types for Assay ALA3858378
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 438.81 | 4.84 | 4.84 |
| 439.80 | 4.23 | 4.23 |
| 437.82 | 5.44 | 5.44 |
| 420.82 | 4.70 | 4.70 |