Basic Information
ID: ALA3858850
Type: Binding
Description: Inhibition of human ERG expressed in HEK293 cells assessed as reduction in maximal tail current at 3 uM and holding potential of -60 mV measured after 5 mins by patch-clamp assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA3858850
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 400.45 | 5.08 | 5.08 |
| 344.89 | 4.69 | 4.69 |
| 464.48 | 5.79 | 5.79 |
| 428.50 | 5.25 | 5.25 |
| 450.46 | 5.36 | 5.36 |
| 432.47 | 5.22 | 5.22 |
| 432.47 | 5.16 | 5.16 |
| 451.44 | 4.30 | 4.30 |
| 444.50 | 4.84 | 4.84 |
| 480.48 | 5.16 | 5.16 |
| 414.48 | 5.08 | 5.08 |
| 450.46 | 5.36 | 5.36 |
| 464.48 | 5.79 | 5.79 |
| 448.92 | 5.73 | 5.73 |
| 414.48 | 5.08 | 5.08 |
| 482.47 | 5.80 | 5.80 |
| 484.35 | 5.33 | 5.33 |
| 466.45 | 5.02 | 5.02 |
| 451.44 | 4.30 | 4.30 |
| 465.47 | 4.69 | 4.69 |