Basic Information
ID: ALA3860286
Type: Binding
Description: Inhibition of post-glutamyl peptide hydrolyzing activity of human 20S proteasome at 50 uM using Cbz-Leu-Leu-Glu-AMC as substrate measured for 10 mins by fluorescence assay relative to control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3860286
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 459.54 | 5.40 | 5.40 |
| 332.36 | 0.70 | 0.70 |
| 331.30 | 1.92 | 1.92 |
| 513.59 | 1.71 | 1.71 |
| 327.38 | 2.58 | 2.58 |
| 462.50 | 3.04 | 3.04 |
| 268.27 | 1.61 | 1.61 |
| 413.47 | 2.00 | 2.00 |
| 334.37 | 0.59 | 0.59 |
| 300.38 | 2.16 | 2.16 |
| 576.65 | 4.98 | 4.98 |
| 285.30 | -2.26 | -2.26 |
| 413.47 | 1.86 | 1.86 |
| 384.52 | 2.92 | 2.92 |
| 354.36 | 1.85 | 1.85 |
| 414.46 | 2.46 | 2.46 |
| 476.53 | 3.48 | 3.48 |
| 492.57 | 1.00 | 1.00 |
| 479.57 | 1.51 | 1.51 |
| 428.49 | 2.85 | 2.85 |
| 293.32 | 0.84 | 0.84 |
| 361.42 | 1.02 | 1.02 |
| 356.40 | 3.74 | 3.74 |
| 300.38 | 3.14 | 3.14 |
| 607.71 | 4.15 | 4.15 |
| 327.38 | -1.44 | -1.44 |
| 414.56 | 3.02 | 3.02 |
| 287.32 | 1.86 | 1.86 |
| 294.35 | 2.78 | 2.78 |
| 302.36 | 1.99 | 1.99 |
| 369.42 | 1.51 | 1.51 |
| 335.40 | 3.41 | 3.41 |
| 296.37 | 2.68 | 2.68 |
| 413.47 | 2.00 | 2.00 |
| 335.38 | 1.51 | 1.51 |
| 455.51 | 1.71 | 1.71 |
| 324.29 | 3.25 | 3.25 |
| 529.59 | 0.23 | 0.23 |
| 497.59 | 2.73 | 2.73 |
| 315.35 | 3.17 | 3.17 |
| 427.50 | 2.25 | 2.25 |
| 294.31 | -0.02 | -0.02 |
| 428.49 | 2.85 | 2.85 |