Basic Information
ID: ALA3864474
Type: Binding
Description: Inhibition of recombinant human N-terminal His6-tagged Keap1 Kelch domain (321 to 609 residues) expressed in Escherichia coli interaction with Nrf2 assessed as displacement of FITC-betaAla-DEETGEF-OH from Keap1 Kelch domain after 30 mins by FP assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3864474
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 835.82 | -3.55 | -3.55 |
| 801.80 | -3.75 | -3.75 |
| 980.98 | -3.66 | -3.66 |
| 809.78 | -4.04 | -4.04 |