Assay Report Card

Basic Information

ID: ALA3866560

Type: Binding

Description: Inhibition of His-sumo-tagged BALB/c mouse thymus histone methyltransferase G9a (969 to 1263 residues) catalytic domain expressed in Escherichia coli BL21 (DE3) using histone H3 (1 to 24 residues) as substrate assessed as reduction in H3K9me2 levels at 10 uM after 1 hr in presence of SAM by MALDI-TOF-mass spectroscopic analysis

Organism: Mus musculus

Strain: BALB/c

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
579.596.976.97