Basic Information
ID: ALA3866781
Type: Binding
Description: Inhibition of GTPgammaS-induced activation of GIRK1/4 (unknown origin) expressed in HEK293 cells assessed as decrease in channel current after 2 mins at -40 mV holding potential by automated patch-clamp electrophysiology assay
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA3866781
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 620.69 | 2.88 | 2.88 |
| 606.67 | 2.63 | 2.63 |
| 755.81 | 3.33 | 3.33 |
| 654.71 | 3.54 | 3.54 |
| 678.73 | 2.25 | 2.25 |