Basic Information
ID: ALA3870777
Type: Binding
Description: Inhibition of recombinant 6His-tagged human calcineurin-alpha expressed in Escherichia coli BL21(DE3/pLysS) assessed as inhibition of calcineurin phosphatase activity by measuring amount of free phosphate at 10 uM preincubated for 20 mins followed by addition of bovine RII phosphopeptide as substrate measured after 30 mins in presence of human calmodulin by malachite green dye-based spectrophotometry relative to DMSO control
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3870777
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1202.63 | ||
| 1218.70 | ||
| 1218.70 | ||
| 1234.77 |