Basic Information
ID: ALA3871085
Type: Binding
Description: Inhibition of recombinant human KLK1 expressed in baculovirus/insect cell expression system using Abz-KLRSSKQ-EDDnp peptide as substrate preincubated for 5 mins followed by substrate addition by FRET assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Kallikrein 1(ALA2319)
Document: ALA3870348
Inhibition of recombinant human KLK1 expressed in baculovirus/insect cell expression system using Abz-KLRSSKQ-EDDnp peptide as substrate preincubated for 5 mins followed by substrate addition by FRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA3871085
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 506.64 | 4.11 | 4.11 |
| 746.95 | 4.53 | 4.53 |
| 702.85 | 5.00 | 5.00 |
| 901.07 | 6.14 | 6.14 |
| 775.00 | 5.14 | 5.14 |
| 750.93 | 5.40 | 5.40 |
| 536.67 | 3.74 | 3.74 |
| 538.66 | 4.18 | 4.18 |
| 686.89 | 5.26 | 5.26 |
| 550.70 | 4.05 | 4.05 |