Basic Information
ID: ALA3875856
Type: Binding
Description: Inhibition of GST-tagged human recombinant DYRK1A expressed in Escherichia coli using RS peptide as substrate incubated for 30 mins in presence of [gamma-33 P] ATP by liquid scintillation counting analysis
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA3875856
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 212.25 | 3.03 | 3.03 |
| 245.28 | 3.63 | 3.63 |
| 275.31 | 3.64 | 3.64 |
| 275.31 | 3.64 | 3.64 |
| 275.31 | 3.64 | 3.64 |
| 275.31 | 3.64 | 3.64 |
| 246.27 | 3.02 | 3.02 |
| 245.29 | 3.63 | 3.63 |
| 261.26 | 3.88 | 3.88 |
| 225.25 | 2.63 | 2.63 |
| 277.71 | 4.39 | 4.39 |
| 242.28 | 4.35 | 4.35 |
| 243.27 | 3.74 | 3.74 |
| 273.30 | 3.75 | 3.75 |
| 273.30 | 3.75 | 3.75 |
| 243.27 | 3.74 | 3.74 |
| 225.25 | 2.63 | 2.63 |
| 243.27 | 3.74 | 3.74 |
| 305.34 | 3.64 | 3.64 |
| 244.26 | 3.14 | 3.14 |
| 244.30 | 4.23 | 4.23 |
| 264.29 | 2.70 | 2.70 |
| 263.27 | 3.77 | 3.77 |
| 245.28 | 3.52 | 3.52 |
| 245.28 | 3.63 | 3.63 |
| 273.30 | 3.75 | 3.75 |
| 276.30 | 3.03 | 3.03 |
| 321.34 | 2.99 | 2.99 |
| 291.31 | 2.98 | 2.98 |
| 290.33 | 2.92 | 2.92 |
| 303.32 | 3.76 | 3.76 |
| 305.38 | 3.94 | 3.94 |
| 291.31 | 2.98 | 2.98 |
| 303.32 | 3.76 | 3.76 |
| 316.36 | 3.63 | 3.63 |
| 316.32 | 2.95 | 2.95 |
| 279.73 | 4.28 | 4.28 |
| 245.28 | 3.63 | 3.63 |
| 243.27 | 3.74 | 3.74 |
| 305.34 | 3.64 | 3.64 |
| 274.28 | 3.14 | 3.14 |
| 277.33 | 3.34 | 3.34 |
| 289.34 | 3.94 | 3.94 |
| 331.38 | 4.35 | 4.35 |
| 319.36 | 3.51 | 3.51 |
| 273.30 | 3.75 | 3.75 |
| 243.27 | 3.46 | 3.46 |