Basic Information
ID: ALA3880369
Type: Functional
Description: Antagonist activity at recombinant human N-terminal signal peptide/FLAG epitope-tagged VIPR2 expressed in CHO cells co-expressing CAMYEL assessed as inhibition of VIP-induced cAMP accumulation preincubated for 5 mins with luciferin, coelenterazine H followed by VIP addition measured after 5 mins by BRET assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO
Target: Vasoactive intestinal polypeptide receptor 2(ALA4532)
Document: ALA3879914
Antagonist activity at recombinant human N-terminal signal peptide/FLAG epitope-tagged VIPR2 expressed in CHO cells co-expressing CAMYEL assessed as inhibition of VIP-induced cAMP accumulation preincubated for 5 mins with luciferin, coelenterazine H followed by VIP addition measured after 5 mins by BRET assay: 38
Activity Charts
Bioactivity
Activity Types for Assay ALA3880369
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 536.65 | 2.55 | 2.55 |