Inhibition of human CDS1 using N-terminal biotin labeled SGLYRSPSMPENLNRPR as substrate in presence of [gamma-33P]-ATP after 3 hrs by scintillation co...

Basic Information

ID: ALA3882743

Type: Binding

Description: Inhibition of human CDS1 using N-terminal biotin labeled SGLYRSPSMPENLNRPR as substrate in presence of [gamma-33P]-ATP after 3 hrs by scintillation counting method

Format: BAO_0000357

Organism: Homo sapiens

Target: Serine/threonine-protein kinase Chk2(ALA2527)

Document: ALA3882723

Inhibition of human CDS1 using N-terminal biotin labeled SGLYRSPSMPENLNRPR as substrate in presence of [gamma-33P]-ATP after 3 hrs by scintillation counting method: 38

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA3882743

IC50

Total(57)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
297.31	1.70	1.70
311.34	2.09	2.09
337.38	2.62	2.62
351.41	3.01	3.01
336.40	2.41	2.41
412.49	3.98	3.98
364.45	3.19	3.19
336.40	2.46	2.46
338.41	2.66	2.66
378.48	3.58	3.58
336.40	2.46	2.46
350.42	2.80	2.80
350.42	2.71	2.71
350.42	2.71	2.71
440.55	4.62	4.62
454.57	4.93	4.93
470.57	4.63	4.63
474.99	5.27	5.27
509.44	5.93	5.93
440.55	4.62	4.62
454.57	4.93	4.93
470.57	4.63	4.63
474.99	5.27	5.27
509.44	5.93	5.93
454.57	5.15	5.15
468.60	5.46	5.46
484.60	5.16	5.16
489.02	5.81	5.81
523.46	6.46	6.46
454.57	5.01	5.01
468.60	5.32	5.32
484.60	5.02	5.02
489.02	5.66	5.66
523.46	6.32	6.32
454.53	4.26	4.26
468.56	4.79	4.79
468.56	4.65	4.65
378.43	2.72	2.72
392.46	2.97	2.97
392.46	2.97	2.97
406.49	3.50	3.50
406.49	3.36	3.36
364.45	3.24	3.24
450.54	4.35	4.35
338.41	2.66	2.66
464.57	4.89	4.89
378.43	2.72	2.72
365.43	3.26	3.26
460.97	5.03	5.03
364.45	3.10	3.10
426.52	4.37	4.37
426.52	4.37	4.37
436.51	4.11	4.11
365.43	3.26	3.26
436.51	4.11	4.11
464.57	4.74	4.74
450.54	4.35	4.35