Assay Report Card

Basic Information

ID: ALA3887934

Type: Binding

Description: Competitive Binding Assay (KINOMEscan): For the competitive binding assay, test compounds were screened at 10 uM against 70 diverse kinase targets for competitive binding using the KINOMEscan technology (Ambit Biosciences) (Karaman, et al. (2008) Nature biotechnology 26:127-132). 11-point Kd curves were determined for hits identified during the initial screen.

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
459.465.125.12