Assay Report Card

Basic Information

ID: ALA3999512

Type: Binding

Description: Inverse agonist activity at GAL4-DNA binding domain-fused human ERRalpha ligand binding domain expressed in African green monkey CV1 cells assessed as decrease in receptor transcriptional activity at 10 uM after 45 hrs by luciferase reporter gene assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
417.555.065.06
387.525.705.70
459.595.285.28
473.615.535.53
374.445.015.01
443.596.176.17
415.586.346.34
445.565.245.24
388.465.265.26
431.585.315.31
401.555.955.95
459.595.495.49