Basic Information
ID: ALA4008765
Type: Binding
Description: Inhibition of recombinant human KDM1A/CoREST complex expressed in Escherichia coli using biotinylated H3K4me1 peptide as substrate preincubated for 10 mins with enzyme followed by substrate addition measured after 1 hr by TR-FRET HTS assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4008765
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 439.47 | 3.46 | 3.46 |
| 300.38 | 3.64 | 3.64 |
| 272.39 | 2.46 | 2.46 |
| 356.77 | 5.07 | 5.07 |