Assay Report Card

Basic Information

ID: ALA4009364

Type: ADME

Description: Inhibition of recombinant human matriptase (596 to 855 residues) expressed in Escherichia coli using Boc-Gln-Ala-ArgAMC as substrate measured for 1200 mins by fluorescence assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
716.862.082.08
754.871.391.39
683.884.124.12
814.973.823.82
651.833.243.24
700.872.372.37
685.852.842.84
775.985.315.31
697.914.514.51
697.914.514.51
676.873.183.18
683.884.264.26
809.995.615.61
697.914.514.51
771.932.122.12
770.942.722.72
685.852.842.84
796.912.072.07
685.853.433.43
780.912.372.37
729.954.414.41
697.914.514.51
735.313.023.02
683.884.124.12
697.914.514.51
669.853.873.87
803.953.143.14
701.853.143.14
697.914.514.51