Assay Report Card

Basic Information

ID: ALA4009657

Type: Binding

Description: Inhibition of PDK1 in human A549 cells assessed as reduction in phosphorylation of PDHE1 at S232 residue at 1 uM after 24 hrs by chemiluminescence/femtochemiluminescence method

Organism: Homo sapiens

Cell type: A549

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
380.633.163.16
384.570.320.32
440.590.690.69
412.621.631.63
352.572.382.38
412.621.631.63
352.572.382.38
440.682.412.41
468.641.471.47