Basic Information
ID: ALA4009735
Type: Binding
Description: Inhibition of mouse glutaminyl cyclase assessed as reduction in conversion of H-Gln-AMC hydrobromide to pGlu-AMC preincubated with substrate for 10 mins followed by enzyme addition by pGAPase coupled fluorometry
Format: BAO_0000357
Organism: Mus musculus
Target: Glutaminyl-peptide cyclotransferase(ALA4105900)
Document: ALA4007443
Inhibition of mouse glutaminyl cyclase assessed as reduction in conversion of H-Gln-AMC hydrobromide to pGlu-AMC preincubated with substrate for 10 mins followed by enzyme addition by pGAPase coupled fluorometry: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4009735
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 334.45 | 2.59 | 2.59 |
| 468.63 | 3.96 | 3.96 |