Basic Information
ID: ALA4011255
Type: Binding
Description: Antagonist activity at human P2Y12 receptor expressed in CHO cells assessed as inhibition of 2-MeSADP-induced beta-arrestin translocation preincubated for 30 mins followed by 2-MeSADP addition measured after 90 mins by luminescence-based topcount method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4011255
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 416.39 | 3.03 | 3.03 |
| 446.42 | 3.05 | 3.05 |
| 552.61 | 5.80 | 5.80 |
| 552.61 | 5.80 | 5.80 |
| 539.57 | 4.72 | 4.72 |
| 552.61 | 5.80 | 5.80 |