Basic Information
ID: ALA4011335
Type: Binding
Description: Displacement of [125I]N6-(4-amino-3-iodobenzyl)adenosine-5'-N-methyluronamide from human A3AR expressed in HEK293T cells pre-incubated for 10 mins before radioligand addition and measured 90 mins after radioligand addition by micro beta scintillation counting analysis relative to control
Organism: Homo sapiens
Cell type: HEK-293T
Activity Charts
Bioactivity
Activity Types for Assay ALA4011335
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 459.92 | 1.44 | 1.44 |
| 550.04 | 3.05 | 3.05 |
| 502.00 | 2.61 | 2.61 |
| 504.37 | 1.55 | 1.55 |
| 457.94 | 1.62 | 1.62 |
| 487.97 | 2.22 | 2.22 |
| 445.89 | 1.35 | 1.35 |
| 472.95 | 2.43 | 2.43 |
| 516.02 | 2.85 | 2.85 |
| 487.97 | 0.34 | 0.34 |
| 476.95 | 1.13 | 1.13 |
| 536.01 | 3.01 | 3.01 |
| 448.89 | 0.35 | 0.35 |
| 449.88 | 0.77 | 0.77 |
| 473.94 | 1.83 | 1.83 |
| 564.07 | 3.44 | 3.44 |
| 518.39 | 1.94 | 1.94 |
| 487.97 | 2.22 | 2.22 |
| 556.09 | 3.78 | 3.78 |