Inhibition of recombinant human N-terminal GST-fused PAK4 (1 to 591 residues) expressed in baculovirus expression system using S2 as substrate measure...

Basic Information

ID: ALA4012135

Type: Binding

Description: Inhibition of recombinant human N-terminal GST-fused PAK4 (1 to 591 residues) expressed in baculovirus expression system using S2 as substrate measured after 40 mins by HTRF assay

Format: BAO_0000019

Organism: Homo sapiens

Target: Serine/threonine-protein kinase PAK 4(ALA4482)

Document: ALA4011593

Inhibition of recombinant human N-terminal GST-fused PAK4 (1 to 591 residues) expressed in baculovirus expression system using S2 as substrate measured after 40 mins by HTRF assay: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA4012135

IC50

Total(24)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
466.54	4.35	4.35
490.64	4.53	4.53
437.48	5.52	5.52
454.93	5.43	5.43
449.52	5.39	5.39
449.52	5.39	5.39
532.83	6.80	6.80
453.94	6.04	6.04
498.39	6.15	6.15
453.94	6.04	6.04
453.94	6.04	6.04
498.39	6.15	6.15
449.52	5.39	5.39
453.94	6.04	6.04
488.38	6.69	6.69
453.94	6.04	6.04
449.52	5.39	5.39
467.96	6.35	6.35
437.48	5.52	5.52
419.49	5.39	5.39
468.95	5.66	5.66
453.94	6.04	6.04
454.93	5.43	5.43
419.49	5.39	5.39