Assay Report Card

Basic Information

ID: ALA4013145

Type: Binding

Description: Antagonist activity at rat alpha6/alpha3beta4 nACHR expressed in xenopous laevis oocyte assessed as inhibition of ACh induced channel current after 5 mins at -70 mV holding potential by two electrode voltage clamp method relative to alpha-conotoxin

Organism: Rattus norvegicus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1487.85
1461.76
1546.87
1487.85
1505.77
1517.87
1487.85
1455.78
1545.93
1553.86