Assay Report Card

Basic Information

ID: ALA4014239

Type: Binding

Description: Intrinsic activity at human GPR34 expressed in HEK293 cells co-transfected with AP-TGFalpha/chimeric Galphaq/i1 assessed as induction of AP-TGFalpha release after 1 hr relative to O-(Hydroxy(((2R,3R)-2-(((3-(2-((3-phenoxybenzyl)oxy)phenyl)- propanoyl)oxy)methyl)tetrahydro-2H-pyran-3-yl)oxy)phosphoryl)- L-serine

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
523.604.474.47
629.604.634.63
587.564.784.78
573.544.474.47
587.564.784.78
629.645.775.77
649.636.146.14
705.747.437.43
587.564.784.78
725.737.807.80