Assay Report Card

Basic Information

ID: ALA4015189

Type: Binding

Description: Inhibition of human TRPV1 expressed in HEK293 cells assessed as decrease in capsaicin-evoked increase in intracellular calcium level at 22 uM preincubated for 2 mins followed by capsaicin addition measured for 2.5 mins by Fluo8-AM dye-based fluorescence assay relative to control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
448.454.774.77