Assay Report Card

Basic Information

ID: ALA4015205

Type: Binding

Description: Selectivity ratio of EC50 for mouse TRPC6 expressed in HEK293 cells co-expressing Gq11-PLCbeta fused M5 receptor assessed as increase in intracellular calcium level to EC50 for human TRPC3 expressed in HEK293 cells assessed as induction of membrane depolarization in presence of 0.5 mM Ca2+

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
448.454.774.77