Assay Report Card

Basic Information

ID: ALA4017304

Type: Binding

Description: Inhibition of full length HIF-PHD1 (unknown origin) expressed in baculovirus infected sf9 cells using DLDLEMLAPYIPMDDDFQL/2-Oxoglutarate as substrate preincubated for 15 mins followed by substrate addition measured after 30 mins by UPLC-MS analysis

Organism: Homo sapiens

Activity Charts

Bioactivity

Activity Types for Assay ALA4017304

IC50

Total(66)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
221.22	1.66	1.66
209.25	2.70	2.70
225.25	2.40	2.40
225.25	2.40	2.40
254.68	2.92	2.92
234.26	2.58	2.58
252.25	2.72	2.72
221.22	1.66	1.66
256.21	2.55	2.55
277.29	2.23	2.23
250.26	2.28	2.28
264.12	3.70	3.70
234.26	2.58	2.58
229.67	3.05	3.05
277.29	2.23	2.23
235.25	1.85	1.85
249.28	2.16	2.16
234.26	2.58	2.58
248.29	2.83	2.83
234.26	2.58	2.58
238.22	2.41	2.41
210.20	1.86	1.86
254.68	2.92	2.92
234.26	2.58	2.58
210.20	0.79	0.79
213.24	1.08	1.08
256.21	2.55	2.55
195.22	2.40	2.40
277.29	2.23	2.23
229.67	3.05	3.05
235.25	1.85	1.85
291.31	2.53	2.53
213.22	2.54	2.54
227.27	1.47	1.47
220.24	2.27	2.27
225.25	2.40	2.40
288.23	3.29	3.29
235.25	1.85	1.85
222.21	1.06	1.06
252.25	2.72	2.72
226.26	2.33	2.33
288.23	3.29	3.29
238.22	2.41	2.41
209.25	2.70	2.70
238.22	2.41	2.41
238.22	2.41	2.41
222.21	1.06	1.06
248.29	2.88	2.88
263.30	2.70	2.70
277.29	2.23	2.23
256.21	2.55	2.55
234.26	2.58	2.58
210.20	0.79	0.79
264.12	3.70	3.70
239.28	1.47	1.47
229.67	3.05	3.05
263.30	2.33	2.33
213.22	2.54	2.54
220.24	2.27	2.27
228.26	0.33	0.33
252.25	2.72	2.72
222.21	1.06	1.06
264.12	3.70	3.70
263.30	2.33	2.33
235.25	1.85	1.85
213.22	2.54	2.54