ID: ALA4024931
Type: Binding
Description: Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as substrate pretreated for 60 mins followed by substrate addition after 1 hr by ADP-Glo luminescence assay
Format: BAO_0000219
Organism: Homo sapiens
Target: Tyrosine-protein kinase BTK(ALA5251)
Document: ALA4024706
Inhibition of full length recombinant human N-terminal His tagged BKT expressed in baculovirus infected Sf9 insect cells using poly (Glu,Tyr)4:1 as substrate pretreated for 60 mins followed by substrate addition after 1 hr by ADP-Glo luminescence assay: 1
Bioactivity
Activity Types for Assay ALA4024931
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
440.51 | 4.22 | 4.22 |
499.51 | 4.77 | 4.77 |
560.54 | 6.18 | 6.18 |
423.45 | 4.25 | 4.25 |
633.75 | 6.08 | 6.08 |
708.86 | 6.06 | 6.06 |
647.78 | 6.25 | 6.25 |
659.67 | 5.97 | 5.97 |
513.64 | 4.27 | 4.27 |
605.74 | 6.48 | 6.48 |
675.83 | 7.03 | 7.03 |
659.67 | 5.97 | 5.97 |
645.76 | 5.83 | 5.83 |
548.69 | 7.09 | 7.09 |
622.73 | 4.92 | 4.92 |
591.67 | 4.95 | 4.95 |
746.91 | 7.47 | 7.47 |
635.68 | 4.68 | 4.68 |
621.69 | 4.96 | 4.96 |
605.70 | 5.26 | 5.26 |
513.64 | 3.95 | 3.95 |
631.78 | 7.01 | 7.01 |
647.78 | 6.25 | 6.25 |
660.82 | 6.17 | 6.17 |
578.71 | 6.13 | 6.13 |
447.50 | 4.01 | 4.01 |
647.78 | 6.25 | 6.25 |
670.21 | 6.30 | 6.30 |
673.69 | 6.28 | 6.28 |
681.75 | 4.98 | 4.98 |
662.79 | 5.80 | 5.80 |
649.79 | 6.48 | 6.48 |
619.72 | 5.52 | 5.52 |
634.74 | 5.02 | 5.02 |
649.70 | 4.72 | 4.72 |
661.80 | 6.38 | 6.38 |
660.77 | 5.55 | 5.55 |
527.67 | 4.70 | 4.70 |
592.70 | 6.57 | 6.57 |
676.77 | 4.79 | 4.79 |
651.79 | 5.89 | 5.89 |
513.64 | 3.95 | 3.95 |
651.72 | 4.97 | 4.97 |
513.64 | 4.27 | 4.27 |
617.75 | 6.67 | 6.67 |
621.69 | 4.96 | 4.96 |
648.76 | 5.14 | 5.14 |
534.66 | 6.78 | 6.78 |
648.76 | 5.14 | 5.14 |