Basic Information
ID: ALA4029946
Type: Binding
Description: Positive allosteric modulation at human GABA-B1 expressed in CHO-K1 cell membranes co-expressing rat GABA-B2 assessed as potentiation of GABA-induced reduction in [3H]-CGP62349 binding to GABA-B1 receptor at 0.3 uM measured after 20 mins in presence of 0.3 uM GABA by scintillation counting method relative to 100 uM GABA alone
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4029946
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 337.45 | 3.82 | 3.82 |