ID: ALA4031697
Type: Binding
Description: Inhibition of human BGT1 expresses in tsA201 cells assessed as reduction in [3H]GABA uptake after 3 mins by scintillation counting method
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4031697
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
103.12 | -0.19 | -0.19 |
354.45 | 3.10 | 3.10 |
344.46 | 4.23 | 4.23 |
294.40 | 3.08 | 3.08 |
338.45 | 3.48 | 3.48 |
363.29 | 4.39 | 4.39 |
364.28 | 3.78 | 3.78 |
364.28 | 3.78 | 3.78 |
273.16 | 2.48 | 2.48 |
338.41 | 2.81 | 2.81 |
408.29 | 4.30 | 4.30 |
364.28 | 3.78 | 3.78 |
391.30 | 4.07 | 4.07 |
489.18 | 4.99 | 4.99 |
389.33 | 4.90 | 4.90 |
451.33 | 4.84 | 4.84 |
413.35 | 5.54 | 5.54 |
287.19 | 2.82 | 2.82 |
387.31 | 3.53 | 3.53 |
315.24 | 3.60 | 3.60 |
331.20 | 2.27 | 2.27 |
340.25 | 3.49 | 3.49 |
311.21 | 2.82 | 2.82 |
362.39 | 4.10 | 4.10 |
364.28 | 3.78 | 3.78 |
312.39 | 3.22 | 3.22 |
260.38 | 2.42 | 2.42 |
421.32 | 4.17 | 4.17 |
388.30 | 4.26 | 4.26 |
414.34 | 4.94 | 4.94 |
388.30 | 4.26 | 4.26 |
301.22 | 3.21 | 3.21 |
408.29 | 4.30 | 4.30 |