Basic Information
ID: ALA4040125
Type: Binding
Description: Inhibition of human NaV1.7 expressed in HEK cells assessed as half inactivation potential at -120 mV holding potential by automated patch clamp method
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4040125
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 471.95 | 4.66 | 4.66 |
| 504.48 | 4.48 | 4.48 |
| 504.48 | 4.48 | 4.48 |
| 472.94 | 4.06 | 4.06 |
| 511.34 | 5.66 | 5.66 |
| 494.34 | 4.92 | 4.92 |
| 530.91 | 6.00 | 6.00 |
| 499.38 | 5.58 | 5.58 |
| 465.92 | 4.32 | 4.32 |
| 458.91 | 4.05 | 4.05 |
| 541.06 | 5.00 | 5.00 |
| 472.94 | 4.06 | 4.06 |
| 500.36 | 4.98 | 4.98 |
| 531.90 | 5.40 | 5.40 |
| 484.95 | 4.30 | 4.30 |
| 500.36 | 5.15 | 5.15 |
| 457.92 | 4.65 | 4.65 |
| 552.03 | 5.41 | 5.41 |
| 504.48 | 4.48 | 4.48 |
| 473.93 | 3.63 | 3.63 |
| 538.00 | 5.02 | 5.02 |
| 458.91 | 4.05 | 4.05 |
| 483.91 | 4.46 | 4.46 |
| 533.92 | 5.52 | 5.52 |
| 506.49 | 4.72 | 4.72 |
| 538.99 | 4.41 | 4.41 |
| 534.90 | 4.91 | 4.91 |