Assay Report Card

Basic Information

ID: ALA4040600

Type: Binding

Description: Inhibition of recombinant human N-terminal GST-tagged IKKalpha (1 to 745 residues) expressed in baculovirus expression system using biotinylated IkBalpha as substrate after 60 mins by DELFIA

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
174.17-0.01-0.01
272.311.131.13
217.281.531.53
313.341.481.48
218.22-0.18-0.18
299.303.303.30
328.361.451.45
253.242.222.22
278.281.181.18
244.260.250.25
321.37-0.33-0.33
274.311.271.27
264.292.022.02
250.262.162.16
247.301.261.26
328.360.990.99
314.330.730.73
278.281.181.18
188.190.450.45
300.371.541.54
319.371.741.74
244.26-0.02-0.02
168.591.191.19
253.242.222.22
258.280.370.37
256.312.162.16
278.281.181.18
290.28-1.32-1.32
258.280.370.37
265.281.571.57
251.251.781.78
299.321.141.14
265.281.571.57
314.330.730.73
287.330.160.16
290.330.350.35
251.251.781.78
293.291.251.25
257.300.160.16
242.291.401.40
265.281.571.57
289.320.850.85
274.28-0.29-0.29
193.601.071.07
301.35-0.08-0.08
329.350.800.80
231.302.282.28
404.463.193.19
270.342.182.18
228.261.231.23
287.33-0.47-0.47
253.242.222.22
314.330.730.73
235.252.082.08
251.251.781.78
244.26-0.02-0.02