Assay Report Card

Basic Information

ID: ALA4041394

Type: Functional

Description: Antagonist activity at mouse melanocortin receptor 4 expressed in HEK293 cells assessed as inhibition of NDP-MSH-induced cAMP accumulation after 2 hrs by AlphaScreen assay

Organism: Mus musculus

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
977.14-1.22-1.22
901.04-2.45-2.45
963.11-1.61-1.61
976.190.950.95
1049.25
949.13-1.14-1.14
964.14-0.72-0.72
1043.20
993.14-2.25-2.25
934.11-0.08-0.08
1035.17
948.140.310.31
976.191.091.09
1019.22
1010.21
978.12-0.62-0.62
1034.23
962.170.560.56
1053.23
1021.15
992.15-0.23-0.23
950.11-1.11-1.11
949.13-1.14-1.14
1000.17