Basic Information
ID: ALA4043421
Type: Binding
Description: Inhibition of recombinant human N-terminal His6-tagged BRD4 bromodomain 1 expressed in Escherichia coli BL21(DE3) using biotinylated histone peptide as substrate after 60 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4043421
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 513.62 | 5.68 | 5.68 |
| 532.65 | 6.94 | 6.94 |
| 516.64 | 5.68 | 5.68 |