Assay Report Card

Basic Information

ID: ALA4043645

Type: Binding

Description: Inhibition of GRK2 in isoproterenol-stimulated C57/BL6 mouse cardiomyocytes assessed as increase in contractility by measuring cell shortening at 1 uM pretreated for 10 mins followed by beta-AR agonist isoproterenol addition for 2 mins

Organism: Mus musculus

Strain: C57/BL6

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
365.372.972.97
463.513.653.65