Assay Report Card

Basic Information

ID: ALA4043794

Type: Binding

Description: Inhibition of human phosphorylated ABL1 E255K mutant (S229 to K512 residues) expressed in HEK293 cells assessed as residual activity at 1000 nM after 30 mins by Kinomescan method relative to control

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
658.565.745.74