Basic Information
ID: ALA4046326
Type: Binding
Description: Inhibition of human OCT2 expressed in HEK293 cells assessed as decrease in uptake of substrate [3H]MPP+ after 1 min by liquid scintillation counting method
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA4046326
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 169.62 | 1.65 | 1.65 |
| 135.17 | 0.99 | 0.99 |
| 149.20 | 1.30 | 1.30 |
| 169.62 | 1.65 | 1.65 |
| 225.29 | 2.58 | 2.58 |
| 214.07 | 1.75 | 1.75 |
| 153.16 | 1.13 | 1.13 |
| 191.28 | 1.89 | 1.89 |
| 261.07 | 1.20 | 1.20 |