Basic Information
ID: ALA4047930
Type: Binding
Description: Inhibition of human VAP-1 expressed in CHO cells preincubated for 20 mins followed by [14C]-benzylamine addition measured after 1 hr by scintillation spectrometric analysis
Format: BAO_0000219
Organism: Homo sapiens
Target: Amine oxidase, copper containing(ALA3437)
Document: ALA4043269
Inhibition of human VAP-1 expressed in CHO cells preincubated for 20 mins followed by [14C]-benzylamine addition measured after 1 hr by scintillation spectrometric analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4047930
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 511.53 | 1.11 | 1.11 |
| 470.83 | 1.11 | 1.11 |
| 520.50 | 1.41 | 1.41 |
| 506.47 | 1.10 | 1.10 |
| 399.33 | 1.40 | 1.40 |
| 522.49 | 1.67 | 1.67 |
| 886.97 | 0.65 | 0.65 |
| 934.82 | 1.38 | 1.38 |
| 410.84 | 1.24 | 1.24 |
| 523.47 | 1.92 | 1.92 |
| 491.50 | 0.90 | 0.90 |
| 463.80 | 1.53 | 1.53 |
| 538.49 | 1.55 | 1.55 |
| 427.38 | 1.12 | 1.12 |
| 463.80 | 1.53 | 1.53 |
| 399.33 | 1.40 | 1.40 |
| 519.52 | 1.02 | 1.02 |
| 523.47 | 1.92 | 1.92 |
| 537.50 | 2.39 | 2.39 |
| 447.30 | 1.24 | 1.24 |
| 463.75 | 1.75 | 1.75 |
| 463.80 | 1.53 | 1.53 |
| 868.81 | 1.61 | 1.61 |
| 490.47 | 0.53 | 0.53 |